Smyth, D . G . ( 1967 ) Carbamylation of amino and tyrosine hydroxyl groups : preparation of an inhibitor of oxytocin with no intrinsic activity on the isolated uterus.
12.
"' EVT-201 "'is a benzodiazepine ? 5 subunits and significantly less intrinsic activity in comparison to currently-marketed benzodiazepines and the Z-drugs.
13.
Moreover, due to partial agonism of the KOR, where it appears to possess significantly greater intrinsic activity relative to the MOR, diprenorphine can produce sedation as well as, in humans, hallucinations.
14.
However, in the presence of full agonists like testosterone or dihydrotestosterone ( DHT ), due to its lower intrinsic activity in comparison, it has antagonistic effects, and can behave more like an antiandrogen.
15.
However, due to its lower intrinsic activity in comparison, in the presence of full agonists like testosterone or dihydrotestosterone ( DHT ), 4-androstenediol has antagonistic actions, behaving more like an antiandrogen.
16.
An important accomplishment of Ari�ns was the establishment of experiments on isolated organs instead of the living animal ( " ex vivo " ), which quickly and reproducibly delivered data on the affinity and intrinsic activity of test substances.
17.
Taking a more sophisticated approach, receptor reserve is an integrative measure of the response-inducing capacity of an agonist ( in some receptor models it is termed intrinsic efficacy or intrinsic activity ) and of the signal amplification capacity of the corresponding receptor ( and its downstream signaling pathways ).
18.
"' Levallorphan "'( antagonist of the ?-opioid receptor ( MOR ) and as an agonist of the ?-opioid receptor ( KOR ), and as a result, blocks the effects of stronger agents with greater intrinsic activity such as morphine whilst simultaneously producing analgesia.
19.
Thus, the production of hepoxilins from 12 ( S )-HpETE may result from the intrinsic activity of platelet or leukocyte type 12-LOX's, require eLOX3, or even result from 12 ( " S " )-HpETE spontaneous ( and perhaps artifactual ) decomposition during isolation.
20.
DPN is a racemic mixture of two enantiomers, ( R )-DPN and ( S )-DPN . Relative to ( R )-DPN, ( S )-DPN has between 3-and 7-fold higher affinity for ER? and appears to have higher intrinsic activity in activating ER?.
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